Description
Catalogue Number | IM046081 |
CAS No. | 1346599-72-1 |
Alternate CAS No. | unlabelled: 33671-46-4 |
Chemical Name | Clotiazepam-13C,d3 |
Synonyms | 5-(o-Chlorophenyl)-7-ethyl-1,3-dihydro-1-(methyl-13C,d3)-2H-thieno[2,3-e]-1,4-diazepin-2-one; Clozan-13C,d3; Rize-13C,d3; Rizen-13C,d3; 5-(o-Chlorophenyl)-7-ethyl-1-(methyl-13C,d3)-1,2-dihydro-3H-thieno[2,3-e][1,4]diazepin-2-one; Tienor-13C,d3; Trecalmo-13C,d3; Veratran-13C,d3; Y 6047-13C,d3; 1-(Methyl-13C,d3)-5-o-chlorophenyl-7-ethyl-1,2-dihydro-3H-thieno[2,3-e][1,4]diazepin-2-one; |
Molecular Formula | C₁₅¹³CH₁₂D₃ClN₂OS |
Molecular Weight | 322.83 |
Appearance | Off-White to Pale Yellow Solid |
Melting Point | 106-107°C |
Storage | -20°C |
Solubility | DMSO (Slightly), Methanol (Slightly) |
Applications | A labelled thienodiazepine derivative that possesses anxiolytic, skeletal muscle relaxant anticonvulsant, sedative properties as well as contributing to siginificant increase stage 2 NREM sleep. It binds to benzodiazepine site of the GABAA receptor where it acts as a full agonist resulting in enhanced GABA inhibitory effect at the GABAA receptor.Controlled Substance. |
Category | Standards; Isotopic Labeled Analogues; Enzyme Activators and Inhibitors; Pharmaceutical/API Drug Impurities/Metabolites; Controlled Substances and Drugs of Abuse for Forensic Testing; Sedatives; Benzodiazepines; |
Note: All Products are stable to be shipped at room temperature, unless otherwise specified.